Catalytic one-pot synthesis of 4-(hetero)aryl substituted 5-(2-oxoethyl) oxazol-2(3H)-ones by coupling–isomerization–elimination (CIE) sequence-Reference-Cited by-同舟云学术

Catalytic one-pot synthesis of 4-(hetero)aryl substituted 5-(2-oxoethyl) oxazol-2(3H)-ones by coupling–isomerization–elimination (CIE) sequence

Published:2016 Issue:7 Volume:3 Page:887-896
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Görgen née Boersch Christina¹²³⁴⁵,Lutsenko Kiril¹²³⁴⁵,Merkul Eugen¹²³⁴⁵,Frank Walter⁶²³⁴⁵,Müller Thomas J. J.¹²³⁴⁵

Affiliation:

1. Institut für Organische Chemie und Makromolekulare Chemie

2. Heinrich-Heine-Universität Düsseldorf

3. Universitätsstraße 1

4. 40225 Düsseldorf

5. Germany

6. Institut für Anorganische Chemie und Strukturchemie

Abstract

4-(Hetero)aryl substituted 5-(2-oxoethyl) oxazol-2(3H)-ones are readily prepared in a one-pot fashion by a coupling–isomerization–elimination (CIE) sequence fromN-Boc protected 1-aryl propargyl carbamates and acid chlorides.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/QO/C6QO00138F

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3. Synthesis and Herbicidal Activities of 4-Substituted 3-Aryl-5-tert-butyl-4-oxazolin-2-ones

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