Synthesis and 18F-radiolabeling of thymidine AMBF3 conjugates-Reference-Cited by-同舟云学术

Synthesis and 18F-radiolabeling of thymidine AMBF3 conjugates

Published:2020 Issue:5 Volume:11 Page:569-576
ISSN:2632-8682
Container-title:RSC Medicinal Chemistry
language:en
Short-container-title:RSC Med. Chem.

Author:

Wong Antonio A. W. L.¹²³⁴^ORCID,Lozada Jerome¹²³⁴,Lepage Mathieu L.¹²³⁴^ORCID,Zhang Chengcheng⁵⁶³⁷,Merkens Helen⁵⁶³⁷,Zeisler Jutta⁵⁶³⁷,Lin Kuo-Shyan⁵⁶³⁷^ORCID,Bénard François⁵⁶³⁷,Perrin David M.¹²³⁴^ORCID

Affiliation:

1. Department of Chemistry

2. University of British Columbia (UBC)

3. Vancouver

4. V6T 1Z1 Canada

5. Department of Molecular Oncology

6. B.C. Cancer Research Centre (BCCRC)

7. V5Z 1L3 Canada

Abstract

One step radiofluorination of two thymidine bioconjugates for positron emission tomography (PET) imaging; proof concept with clinical-grade ¹⁸F-labeling and preliminary mouse images.

Funder

Natural Sciences and Engineering Research Council of Canada

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/MD/D0MD00054J

Reference47 articles.

1. Serum Thymidine Kinase 1 Activity in Solid Tumor (Breast and Colorectal Cancer) Patients Treated With Adjuvant Chemotherapy

2. Imaging proliferation in vivo with [F-18]FLT and positron emission tomography

3. Different Modes of Transport for 3H-Thymidine, 3H-FLT, and 3H-FMAU in Proliferating and Nonproliferating Human Tumor Cells

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