Design, characterization and cellular uptake studies of fluorescence-labeled prototypic cathepsin inhibitors-Reference-Cited by-同舟云学术

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Design, characterization and cellular uptake studies of fluorescence-labeled prototypic cathepsin inhibitors

Published:2015 Issue:41 Volume:13 Page:10310-10323
ISSN:1477-0520
Container-title:Org. Biomol. Chem.
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Kohl Franziska¹²³⁴,Schmitz Janina¹²³⁴⁵,Furtmann Norbert¹²³⁴⁶,Schulz-Fincke Anna-Christina¹²³⁴,Mertens Matthias D.¹²³⁴,Küppers Jim¹²³⁴,Benkhoff Marcel¹²³⁴,Tobiasch Edda⁵⁷⁸,Bartz Ulrike⁵⁷⁸,Bajorath Jürgen⁶⁹¹⁰³¹¹,Stirnberg Marit¹²³⁴,Gütschow Michael¹²³⁴

Affiliation:

1. Pharmaceutical Institute

2. Pharmaceutical Chemistry I

3. University of Bonn

4. D-53121 Bonn, Germany

5. Department of Natural Sciences

6. Department of Life Science Informatics

7. Bonn-Rhein-Sieg University of Applied Sciences

8. D-53359 Rheinbach, Germany

9. B-IT

10. LIMES Program Unit Chemical Biology and Medicinal Chemistry

11. D-53113 Bonn, Germany

Abstract

Cysteine cathepsin inhibition and cellular uptake of a coumarin 343-containing dipeptide nitrile was analyzed.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB01613D

Reference66 articles.

1. Specialized roles for cysteine cathepsins in health and disease

2. Cysteine cathepsins: From structure, function and regulation to new frontiers

3. Development of Nitrile-Based Peptidic Inhibitors of Cysteine Cathepsins

4. Cysteine cathepsin proteases as pharmacological targets in cancer

5. Cathepsin K: a unique collagenolytic cysteine peptidase

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