Synthesis of novel azole-fused quinazolines via one-pot, sequential Ullmann-type coupling and intramolecular dehydrogenative C

Synthesis of novel azole-fused quinazolines via one-pot, sequential Ullmann-type coupling and intramolecular dehydrogenative C–N bonding

Published:2015 Issue:10 Volume:13 Page:2947-2950
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Nandwana Nitesh Kumar¹²³⁴,Pericherla Kasiviswanadharaju¹²³⁴,Kaswan Pinku¹²³⁴,Kumar Anil¹²³⁴

Affiliation:

1. Department of Chemistry

2. Birla Institute of Technology and Science

3. Pilani 333031

4. India

Abstract

An efficient one-pot sequential procedure is described for the synthesis of novel azole-fused quinazolines through Ullmann-type coupling followed by cross dehydrogenative coupling of various azoles with 2-(2-bromophenyl)-1H-imidazole/benzimidazoles.

Funder

Council for Scientific and Industrial Research

Department of Science and Technology, Ministry of Science and Technology

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C4OB02375G

Reference29 articles.

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