Solid-phase synthesis and fluorine-18 radiolabeling of cycloRGDyK-Reference-Cited by-同舟云学术

Solid-phase synthesis and fluorine-18 radiolabeling of cycloRGDyK

Published:2016 Issue:37 Volume:14 Page:8659-8663
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Davis Ryan A.¹²³²⁴,Lau Kevin¹²³²,Hausner Sven H.¹²³²⁴,Sutcliffe Julie L.¹²³²⁴

Affiliation:

1. Radiochemistry Research and Training Facility

2. USA

3. Department of Biomedical Engineering

4. Department of Internal Medicine

Abstract

A rapid, efficient single continuous process for peptide synthesis, cyclization, and radiolabeling on solid-support with a single purification step afforded a high purity radiotracer.

Funder

U.S. Department of Energy

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/OB/C6OB01636G

Reference43 articles.

1. Molecular imaging: current status and emerging strategies

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