Synergetic copper/TEMPO-catalysed benzylic C–H imidation with N-fluorobenzenesulfonimide at room temperature and tandem conversions with alcohols or arenes-Reference-Cited by-同舟云学术

Synergetic copper/TEMPO-catalysed benzylic C–H imidation with N-fluorobenzenesulfonimide at room temperature and tandem conversions with alcohols or arenes

Published:2021 Issue:13 Volume:8 Page:3298-3307
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Shao Zhong¹²³⁴⁵,Wang Fang¹²³⁴⁵,Shi Jingqi¹²³⁴⁵,Ma Lifang¹²³⁴⁵,Li Ziyuan¹²³⁴⁵^ORCID

Affiliation:

1. Department of Pharmaceutical and Biological Engineering

2. School of Chemical Engineering

3. Sichuan University

4. Chengdu 610065

5. China

Abstract

A remote carbamate-directed benzylic C–H imidation with NFSI at room temperature through synergetic CuCl-TEMPO catalysis and tandem alkoxylation or arylation with alcohols or arenes are described.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/QO/D1QO00340B

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3. Design, synthesis and anticancer activities of novel otobain derivatives