A one-pot multicomponent approach to a new series of morphine derivatives and their biological evaluation
Author:
Affiliation:
1. Department of Chemistry
2. Zhejiang Sci-Tech University
3. Hangzhou
4. P. R. China
5. Torrey Pines Institute for Molecular Studies
6. Port St Lucie
7. USA
8. College of Pharmaceutical Science
9. Zhejiang University
Abstract
Morphine derivatives displaying a mixed MOR/DOR biological characteristic were synthesized through a one-pot multicomponent approach.
Funder
National Natural Science Foundation of China
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2017/OB/C7OB01924F
Reference19 articles.
1. A Total Synthesis of (±)-Codeine by 1,3-Dipolar Cycloaddition
2. Selective Opening of Ring C in the Morphine Skeleton by an Unexpected Cleavage of the C5−C6 Bond in Cycloadducts of Thebaine and Acyl Nitroso Compounds
3. 14-Alkoxy- and 14-Acyloxypyridomorphinans: μ Agonist/δ Antagonist Opioid Analgesics with Diminished Tolerance and Dependence Side Effects
4. Opioid Activity of Spinally Selective Analogues of N-Naphthoyl-β-naltrexamine in HEK-293 Cells and Mice
5. Synthesis and Pharmacological Evaluation of 6,7-Indolo/Thiazolo-MorphinansFurther SAR of Levorphanol
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