Comprehensive analysis of loops at protein-protein interfaces for macrocycle design
Author:
Publisher
Springer Science and Business Media LLC
Subject
Cell Biology,Molecular Biology
Link
http://www.nature.com/articles/nchembio.1580.pdf
Reference44 articles.
1. Wells, J.A. & McClendon, C.L. Reaching for high-hanging fruit in drug discovery at protein–protein interfaces. Nature 450, 1001–1009 (2007).
2. Marsault, E. & Peterson, M.L. Macrocycles are great cycles: applications, opportunities, and challenges of synthetic macrocycles in drug discovery. J. Med. Chem. 54, 1961–2004 (2011).
3. Bock, J.E., Gavenonis, J. & Kritzer, J.A. Getting in shape: controlling peptide bioactivity and bioavailability using conformational constraints. ACS Chem. Biol. 8, 488–499 (2013).
4. Vagner, J., Qu, H. & Hruby, V.J. Peptidomimetics, a synthetic tool of drug discovery. Curr. Opin. Chem. Biol. 12, 292–296 (2008).
5. Nowick, J.S. Exploring β-sheet structure and interactions with chemical model systems. Acc. Chem. Res. 41, 1319–1330 (2008).
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