An Internally Controlled Quantitative Target Occupancy Assay for Covalent Inhibitors
Author:
Publisher
Springer Science and Business Media LLC
Subject
Multidisciplinary
Link
http://www.nature.com/articles/s41598-018-32683-w.pdf
Reference14 articles.
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4. Advani, R. H. et al. Bruton tyrosine kinase inhibitor ibrutinib (PCI-32765) has significant activity in patients with relapsed/refractory B-cell malignancies. J Clin Oncol 31, 88–94 (2013).
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