Trapping of ivermectin by a pentameric ligand-gated ion channel upon open-to-closed isomerization
Author:
Publisher
Springer Science and Business Media LLC
Subject
Multidisciplinary
Link
http://www.nature.com/articles/srep42481.pdf
Reference140 articles.
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3. Geary, T. G. Ivermectin 20 years on: maturation of a wonder drug. Trends Parasitol 21, 530–532 (2005).
4. Cully, D. F. et al. Cloning of an avermectin-sensitive glutamate-gated chloride channel from Caenorhabditis elegans. Nature 371, 707–711 (1994).
5. Etter, A., Cully, D. F., Schaeffer, J. M., Liu, K. K. & Arena, J. P. An amino acid substitution in the pore region of a glutamate-gated chloride channel enables the coupling of ligand binding to channel gating. J Biol Chem 271, 16035–16039 (1996).
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