In situ assembly of enzyme inhibitors using extended tethering-Reference-Cited by-同舟云学术

In situ assembly of enzyme inhibitors using extended tethering

Published:2003-02-03 Issue:3 Volume:21 Page:308-314
ISSN:1087-0156
Container-title:Nature Biotechnology
language:en
Short-container-title:Nat Biotechnol

Author:

Erlanson Daniel A.,Lam Joni W.,Wiesmann Christian,Luong Tinh N.,Simmons Robert L.,DeLano Warren L.,Choong Ingrid C.,Burdett Matthew T.,Flanagan W. Michael,Lee Dennis,Gordon Eric M.,O'Brien Tom

Publisher

Springer Science and Business Media LLC

Subject

Biomedical Engineering,Molecular Medicine,Applied Microbiology and Biotechnology,Bioengineering,Biotechnology

Link

http://www.nature.com/articles/nbt786.pdf

Reference39 articles.

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3. Lehn, J.M. & Eliseev, A. Dynamic combinatorial chemistry. Science 291, 2331–2332 (2001).

4. Nicolaou, K.C. et al. Synthesis and biological evaluation of vancomycin dimers with potent activity against vancomycin-resistant bacteria: target-accelerated combinatorial synthesis. Chem. Eur. J. 7, 3824–3843 (2001).

5. Ramstrom, O. & Lehn, J.M. Drug discovery by dynamic combinatorial libraries. Nat. Rev. Drug Disc. 1, 26–32 (2002).

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