USP7 small-molecule inhibitors interfere with ubiquitin binding-Reference-Cited by-同舟云学术

USP7 small-molecule inhibitors interfere with ubiquitin binding

Published:2017-10-18 Issue:7677 Volume:550 Page:534-538
ISSN:0028-0836
Container-title:Nature
language:en
Short-container-title:Nature

Author:

Kategaya Lorna,Di Lello Paola,Rougé Lionel,Pastor Richard,Clark Kevin R.,Drummond Jason,Kleinheinz Tracy,Lin Eva,Upton John-Paul,Prakash Sumit,Heideker Johanna,McCleland Mark,Ritorto Maria Stella,Alessi Dario R.,Trost Matthias,Bainbridge Travis W.,Kwok Michael C. M.,Ma Taylur P.,Stiffler Zachary,Brasher Bradley,Tang Yinyan,Jaishankar Priyadarshini,Hearn Brian R.,Renslo Adam R.,Arkin Michelle R.,Cohen Frederick,Yu Kebing,Peale Frank,Gnad Florian,Chang Matthew T.,Klijn Christiaan,Blackwood Elizabeth,Martin Scott E.,Forrest William F.,Ernst James A.,Ndubaku Chudi,Wang Xiaojing,Beresini Maureen H.,Tsui Vickie,Schwerdtfeger Carsten,Blake Robert A.,Murray Jeremy,Maurer Till,Wertz Ingrid E.

Publisher

Springer Science and Business Media LLC

Subject

Multidisciplinary

Link

http://www.nature.com/articles/nature24006.pdf

Reference30 articles.

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2. Clague, M. J., Heride, C. & Urbé, S. The demographics of the ubiquitin system. Trends Cell Biol. 25, 417–426 (2015)

3. Nicholson, B. & Suresh Kumar, K. G. The multifaceted roles of USP7: new therapeutic opportunities. Cell Biochem. Biophys. 60, 61–68 (2011)

4. Ritorto, M. S. et al. Screening of DUB activity and specificity by MALDI-TOF mass spectrometry. Nat. Commun. 5, 4763 (2014)

5. Hu, M. et al. Crystal structure of a UBP-family deubiquitinating enzyme in isolation and in complex with ubiquitin aldehyde. Cell 111, 1041–1054 (2002)

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