The Pharmacokinetics of a Thiazole Benzenesulfonamide β3-Adrenergic Receptor Agonist and Its Analogs in Rats, Dogs, and Monkeys: Improving Oral Bioavailability

Author:

Stearns Ralph A.,Miller Randy R.,Tang Wei,Kwei Gloria Y.,Tang Frank S.,Mathvink Robert J.,Naylor Elizabeth M.,Chitty Dawn,Colandrea Vincent J.,Weber Ann E.,Colletti Adria E.,Strauss John R.,Keohane Carol Ann,Feeney William P.,Iliff Susan A.,Chiu Shuet-Hing Lee

Publisher

American Society for Pharmacology & Experimental Therapeutics (ASPET)

Subject

Pharmaceutical Science,Pharmacology

Reference26 articles.

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3. Prospects for β3-adrenoreceptor agonists in the treatment of obesity and diabetes.;Arch;Int J Obes,1996

4. Synthesis and SAR of benzyl and phenoxymethylene oxadiazole benzenesulfonamides as selective β3 adrenergic receptor agonist antiobesity agents

5. Human β3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides

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