Berotralstat (BCX7353): Structure-Guided Design of a Potent, Selective, and Oral Plasma Kallikrein Inhibitor to Prevent Attacks of Hereditary Angioedema (HAE)
Author:
Funder
BioCryst
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00511
Reference43 articles.
1. US HAEA Medical Advisory Board 2020 Guidelines for the Management of Hereditary Angioedema
2. Hereditary angioedema: Epidemiology and burden of disease
3. Oral plasma kallikrein inhibitor BCX7353 for treatment of hereditary angioedema
4. Mutational spectrum of the C1INH (SERPING1) gene in patients with hereditary angioedema
5. Treatment of hereditary angioedema: a review (CME)
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