Optimization of the Antibacterial Spectrum and the Developability Profile of the Novel-Class Natural Product Corramycin

Author:

Renard Stephane1,Versluys Stéphanie2,Taillier Thomas3,Dubarry Nelly1,Leroi-Geissler Corinne1,Rey Astrid3,Cornaire Emilie3,Sordello Sylvie2,Carry Jean-Christophe B.4ORCID,Angouillant-Boniface Odile4,Gouyon Thierry4,Thompson Fabienne4,Lebourg Gilles4,Certal Victor4,Balazs Laszlo4,Arranz Esther4,Doerflinger Gilles4,Bretin Francois4,Gervat Vincent4,Brohan Eric4,Kraft Volker5,Boulenc Xavier1,Ducelier Cécile6,Bacqué Eric3,Couturier Cédric3ORCID

Affiliation:

1. Evotec, 40 Avenue Tony Garnier, Lyon 69007, France

2. Evotec, 195, Route d’Espagne, Toulouse 31100, France

3. Evotec, 1541, Avenue Marcel Mérieux, Marcy L’Etoile 69280, France

4. Sanofi, 13 Quai Jules Guesde, Vitry-sur-Seine 94403, France

5. Sanofi-Aventis Deutschland GmbH, Industriepark Hoechst, Frankfurt am Main 65926, Germany

6. Sanofi, 1 Avenue Pierre Brossolette, Chilly-Mazarin 91385, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Reference65 articles.

1. Antibiotics for Emerging Pathogens

2. Antibiotics: from prehistory to the present day

3. Tackling Drug-Resistant Infections Globally: Final Report and Recommendations. Review on Antimicrobial Resistance Chaired by Jim O’Neill, 2016.

4. Global burden of bacterial antimicrobial resistance in 2019: a systematic analysis

5.

Antimicrobial Resistance: Implications and Costs

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