Coupling of an Acyl Migration Prodrug Strategy with Bio-activation To Improve Oral Delivery of the HIV-1 Protease Inhibitor Atazanavir-Reference-Cited by-同舟云学术

Coupling of an Acyl Migration Prodrug Strategy with Bio-activation To Improve Oral Delivery of the HIV-1 Protease Inhibitor Atazanavir

Published:2018-04-25 Issue:9 Volume:61 Page:4176-4188
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Subbaiah Murugaiah A. M.^ORCID,Meanwell Nicholas A.^ORCID,Kadow John F.,Subramani Lakshumanan,Annadurai Mathiazhagan,Ramar Thangeswaran,Desai Salil D.,Sinha Sarmistha,Subramanian Murali,Mandlekar Sandhya,Sridhar Srikanth,Padmanabhan Shweta,Bhutani Priyadeep,Arla Rambabu,Jenkins Susan M.,Krystal Mark R.,Wang Chunfu,Sarabu Ramakanth

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.8b00277

Reference48 articles.

1. Anti-HIV Drug Discovery and Development: Current Innovations and Future Trends

2. Closing the Gap: Increases in Life Expectancy among Treated HIV-Positive Individuals in the United States and Canada

3. Recent Progress in the Development of HIV-1 Protease Inhibitors for the Treatment of HIV/AIDS

4. Investigational protease inhibitors as antiretroviral therapies

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