Design, Synthesis, and Evaluation of New Selective NM23-H2 Binders as c-MYC Transcription Inhibitors via Disruption of the NM23-H2/G-Quadruplex Interaction-Reference-Cited by-同舟云学术

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Design, Synthesis, and Evaluation of New Selective NM23-H2 Binders as c-MYC Transcription Inhibitors via Disruption of the NM23-H2/G-Quadruplex Interaction

Published:2017-08-04 Issue:16 Volume:60 Page:6924-6941
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wang Yu-Qing¹,Huang Zhou-Li¹,Chen Shuo-Bin¹,Wang Chen-Xi¹,Shan Chan¹,Yin Qi-Kun¹,Ou Tian-Miao¹^ORCID,Li Ding¹,Gu Lian-Quan¹,Tan Jia-Heng¹,Huang Zhi-Shu¹^ORCID

Affiliation:

1. School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, People’s Republic of China

Funder

National Natural Science Foundation of China

Natural Science Foundation of Guangdong Province

Guangdong Provincial Key Laboratory of Construction Foundation, Sun Yat-sen University

Science and Technology Development Special Foundation of Guangdong Province

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b00421

Reference37 articles.

1. A SIRT2-Selective Inhibitor Promotes c-Myc Oncoprotein Degradation and Exhibits Broad Anticancer Activity

2. The c-myc oncogene driven by immunoglobulin enhancers induces lymphoid malignancy in transgenic mice

3. Transcriptional Amplification in Tumor Cells with Elevated c-Myc

4. Perturbation of the c-Myc–Max Protein–Protein Interaction via Synthetic α-Helix Mimetics

5. MYC on the Path to Cancer

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1. Synthesis, cytotoxicity study of novel bisacridine derivatives and their interaction with c-myc promoter G-quadruplex/i-motif;Journal of Holistic Integrative Pharmacy;2023-12

2. Development and Characterization of Benzoselenazole Derivatives as Potent and Selective c-MYC Transcription Inhibitors;Journal of Medicinal Chemistry;2023-04-10

3. G-Quadruplexes in c-MYC Promoter as Targets for Cancer Therapy;Biomedicines;2023-03-21

4. Proton‐ and halogen‐induced cyclizations of 2‐(3‐butenyl)quinazolin‐4( 3 H)‐ones in the synthesis of pyrrolo[2,1‐ b ]‐ and pyrrolo[1,2‐ а ]quinazolinone derivatives;Journal of Heterocyclic Chemistry;2022-11-20

5. Design, Synthesis, and Evaluation of New Sugar-Substituted Imidazole Derivatives as Selective c-MYC Transcription Repressors Targeting the Promoter G-Quadruplex;Journal of Medicinal Chemistry;2022-09-19

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