Structure-Enabled Discovery of Novel Macrocyclic Inhibitors Targeting Glutaminase 1 Allosteric Binding Site-Reference-Cited by-同舟云学术

Structure-Enabled Discovery of Novel Macrocyclic Inhibitors Targeting Glutaminase 1 Allosteric Binding Site

Published:2021-04-01 Issue:8 Volume:64 Page:4588-4611
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Xu Xi¹,Wang Jubo¹,Wang Min¹,Yuan Xinyu¹,Li Lei¹,Zhang Chao²,Huang Huidan²,Jing Tian¹,Wang Chenchen¹,Tong Chao¹,Zhou Liwen¹,Meng Ying¹,Xu Pengfei¹,Kou Junping³,Qiu Zhixia¹,Li Zhiyu¹^ORCID,Bian Jinlei¹^ORCID

Affiliation:

1. Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, 24 Tongjiaxiang, Nanjing 210009, P. R. China

2. School of Pharmacy, Wannan Medical College, Wuhu 241002, P. R. China

3. State Key Laboratory of Natural Products, Jiangsu Key Laboratory of TCM Evaluation and Translational Research, Department of Pharmacology of Chinese Material Medical, School of Traditional Chinese Pharmacy, China Pharmaceutical University, Nanjing 211198, P. R. China

Funder

China Pharmaceutical University

China Postdoctoral Science Foundation

Natural Science Foundation of Jiangsu Province

Government of Jiangsu Province

National Natural Science Foundation of China

State Key Laboratory of Drug Research,

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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