Non-rigid Diarylmethyl Analogs of Baloxavir as Cap-Dependent Endonuclease Inhibitors of Influenza Viruses-Reference-Cited by-同舟云学术

Non-rigid Diarylmethyl Analogs of Baloxavir as Cap-Dependent Endonuclease Inhibitors of Influenza Viruses

Published:2020-07-31 Issue:17 Volume:63 Page:9403-9420
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ivashchenko Andrei A.¹²³,Mitkin Oleg D.¹,Jones Jeremy C.⁴,Nikitin Alexander V.¹,Koryakova Angela G.¹,Ryakhovskiy Alexey¹,Karapetian Ruben N.¹,Kravchenko Dmitry V.¹,Aladinskiy Vladimir³^ORCID,Leneva Irina A.⁵,Falynskova Irina N.⁵,Glubokova Ekaterina A.⁵,Govorkova Elena A.⁴,Ivachtchenko Alexandre V.¹²⁶

Affiliation:

1. Chemical Diversity Research Institute, Rabochaya Street 2a, Khimki, Moscow Region 141401, Russia

2. ChemDiv, 6605 Nancy Ridge Drive, San Diego, California 92121, United States

3. Moscow Institute of Physics and Technology (State University), 9 Institutskiy Lane, Dolgoprudny City, Moscow Region 141700, Russia

4. Department of Infectious Diseases, St. Jude Children’s Research Hospital, Memphis, Tennessee 38105, United States

5. I. Mechnikov Research Institute for Vaccines and Sera, 5a Malyy Kazennyy Lane, Moscow 105064, Russia

6. ASAVI LLC, 1835 E. Hallandale Beach Blvd, #442, Hallandale Beach, Florida 33009, United States

Funder

Avisa Pharmaceuticals LLC

Chemical Diversity Research Institute, Khimki, Moscow Region

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c00565

Reference36 articles.

1. A VIRUS OBTAINED FROM INFLUENZA PATIENTS

2. Influenza

3. Influenza Vaccines for the Future

4. Fight Against H1N1 Influenza A Virus: Recent Insights Towards the Development of Druggable Compounds

5. Scientific barriers to developing vaccines against avian influenza viruses

Cited by 18 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Design and synthesis of 7-membered lactam fused hydroxypyridinones as potent metal binding pharmacophores (MBPs) for inhibiting influenza virus PAN endonuclease;European Journal of Medicinal Chemistry;2024-10

2. Solvates and Polymorphs of Baloxavir Marboxil: Crystal Structure and Phase Transformation Study;Crystal Growth & Design;2024-04-08

3. Discovery of a Macrocyclic Influenza Cap-Dependent Endonuclease Inhibitor;Journal of Medicinal Chemistry;2024-02-01

4. Synthesis, intramolecular cyclization, and antinociceptive activity of 4-(het)aryl-2-{[4-(4-chlorophenyl)-3-(ethoxycarbonyl)thiophen-2-yl]amino}-4-oxobut-2-enoic acids;Russian Chemical Bulletin;2023-09

5. Aprotinin—Drug against Respiratory Diseases;International Journal of Molecular Sciences;2023-07-06