Identification of SNAIL1 Peptide-Based Irreversible Lysine-Specific Demethylase 1-Selective Inactivators-Reference-Cited by-同舟云学术

Identification of SNAIL1 Peptide-Based Irreversible Lysine-Specific Demethylase 1-Selective Inactivators

Published:2016-01-04 Issue:4 Volume:59 Page:1531-1544
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Itoh Yukihiro¹,Aihara Keisuke²,Mellini Paolo¹,Tojo Toshifumi¹,Ota Yosuke¹,Tsumoto Hiroki³,Solomon Viswas Raja⁴,Zhan Peng¹,Suzuki Miki¹,Ogasawara Daisuke¹,Shigenaga Akira²,Inokuma Tsubasa²,Nakagawa Hidehiko⁴,Miyata Naoki⁴,Mizukami Tamio⁵,Otaka Akira²,Suzuki Takayoshi¹⁶

Affiliation:

1. Graduate School of Medical Science, Kyoto Prefectural University of Medicine, 1-5 Shimogamohangi-Cho, Sakyo-Ku, Kyoto, 606-0823, Japan

2. Institute of Biomedical Sciences and Graduate School of Pharmaceutical Sciences, Tokushima University, Shomachi, Tokushima 770-8505, Japan

3. Research Team for Mechanism of Aging Tokyo Metropolitan Institute of Gerontology, 35-2 Sakae-Cho, Itabashi-ku, Tokyo 173-0015, Japan

4. Graduate School of Pharmaceutical Sciences, Nagoya City University, 3-1 Tanabe-dori, Mizuho-ku, Nagoya, Aichi 467-8603, Japan

5. Graduate School of Bio-Science, Nagahama Institute of Bio-Science and Technology, 1266 Tamura-cho, Nagahama, Shiga 526-0829, Japan

6. CREST, Japan Science and Technology Agency (JST), 4-1-8 Honcho Kawaguchi, Saitama 332-0012, Japan

Funder

Takeda Science Foundation

Core Research for Evolutional Science and Technology, Japan Science and Technology Agency

Japan Society for the Promotion of Science

Mochida Memorial Foundation for Medical and Pharmaceutical Research

Terumo Foundation for Life Sciences and Arts

Graduate School of Medical Science, Kyoto Prefectural University of Medicine

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01323

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