SLL-627 Is a Highly Selective and Potent κ Opioid Receptor (KOR) Agonist with an Unexpected Nonreduction in Locomotor Activity

Author:

Kong Linghui1ORCID,Shu Xuelian23,Tang Siyuan1,Ye Rongrong4,Sun Huijiao1,Jiang Shuang5,Li Zixiang1,Chai Jingrui2,Fang Yun1,Lan Yinjie1,Yu Linqian1,Xie Qiong1,Fu Wei1ORCID,Wang Yujun2,Li Wei1ORCID,Qiu Zhuibai1,Liu Jinggen2,Shao Liming16ORCID

Affiliation:

1. Department of Medicinal Chemistry, School of Pharmacy, Fudan University, No. 826 Zhangheng Road, Shanghai 201203, China

2. CAS Key Laboratory of Receptor Research and State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences and Collaborative Innovation Center for Brain Science, No. 555 Zuchongzhi Road, Shanghai 201203, China

3. University of Chinese Academy of Sciences, No. 19A Yuquan Road, Beijing 100049, China

4. School of Chemical and Environmental Engineering, Shanghai Institute of Technology, No. 100 Haiquan Road, Shanghai 201418, China

5. School of Pharmacy, Nanjing University of Chinese Medicine, No. 138, Xianlin Road, Nanjing 210023, China

6. State Key Laboratory of Medical Neurobiology, Fudan University, No. 138 Yixueyuan Road, Shanghai 200032, China

Funder

Ministry of Science and Technology of the People's Republic of China

Science and Technology Commission of Shanghai Municipality

National Natural Science Foundation of China

Shenzhen-Hong Kong Institute of Brain Science ? Shenzhen Fundamental Research Institutions

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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