Recent Scaffold Hopping Applications in Central Nervous System Drug Discovery
Author:
Affiliation:
1. School of Chemistry, The University of Sydney, Sydney, NSW 2006, Australia
Funder
National Health and Medical Research Council
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c00969
Reference106 articles.
1. Estimated Research and Development Investment Needed to Bring a New Medicine to Market, 2009-2018
2. “Scaffold-Hopping” by Topological Pharmacophore Search: A Contribution to Virtual Screening
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4. Scaffold-hopping as a strategy to address metabolic liabilities of aromatic compounds
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