Probing the Existence of a Metastable Binding Site at the β2-Adrenergic Receptor with Homobivalent Bitopic Ligands-Reference-Cited by-同舟云学术

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Probing the Existence of a Metastable Binding Site at the β2-Adrenergic Receptor with Homobivalent Bitopic Ligands

Published:2019-07-12 Issue:17 Volume:62 Page:7806-7839
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gaiser Birgit I.¹,Danielsen Mia¹,Marcher-Rørsted Emil¹^ORCID,Røpke Jørgensen Kira¹,Wróbel Tomasz M.¹²^ORCID,Frykman Mikael¹,Johansson Henrik¹,Bräuner-Osborne Hans¹^ORCID,Gloriam David E.¹,Mathiesen Jesper Mosolff¹,Sejer Pedersen Daniel¹^ORCID

Affiliation:

1. Department of Drug Design and Pharmacology, University of Copenhagen, Jagtvej 162, 2100 Copenhagen, Denmark

2. Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University of Lublin, 4A Chodźki 20093 Lublin, Poland

Funder

Lundbeckfonden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b00595

Reference101 articles.

1. Seven-transmembrane receptors

2. Structure-Function of the G Protein–Coupled Receptor Superfamily

3. Strategies to Discover Unexpected Targets for Drugs Active at G Protein–Coupled Receptors

4. The 7 TM G-Protein-Coupled Receptor Target Family

5. The GPCR Network: a large-scale collaboration to determine human GPCR structure and function

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1. Designed dualsteric modulators: A novel route for drug discovery;Drug Discovery Today;2024-10

2. Bitopic Ligands Support the Presence of a Metastable Binding Site at the β₂ Adrenergic Receptor;Journal of Medicinal Chemistry;2024-07-02

3. Mechanistic insights into G-protein coupling with an agonist-bound G-protein-coupled receptor;Nature Structural & Molecular Biology;2024-06-12

4. Allosteric Modulators of Serotonin Receptors: A Medicinal Chemistry Survey;Pharmaceuticals;2024-05-28

5. Multitargeting in cardioprotection: An example of biaromatic compounds;Archiv der Pharmazie;2023-06-22

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