Enantioselective Synthesis of SM-130686 Based on the Development of Asymmetric Cu(I)F Catalysis To Access 2-Oxindoles Containing a Tetrasubstituted Carbon-Reference-Cited by-同舟云学术

Enantioselective Synthesis of SM-130686 Based on the Development of Asymmetric Cu(I)F Catalysis To Access 2-Oxindoles Containing a Tetrasubstituted Carbon

Published:2009-05-06 Issue:20 Volume:131 Page:6946-6948
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Tomita Daisuke¹,Yamatsugu Kenzo¹,Kanai Motomu¹,Shibasaki Masakatsu¹

Affiliation:

1. Graduate School of Pharmaceutical Sciences, The University of Tokyo, Hongo, Bunkyo-ku, Tokyo 113-0033, Japan

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja901995a

Reference32 articles.

1. Oxindole Derivatives as Orally Active Potent Growth Hormone Secretagogues

2. Structure–activity relationships of the oxindole growth hormone secretagogues

3. On an industrial scale, pharmaceuticals that are not derived from natural sources containing chiral tetrasubstituted carbons are almost always produced through resolution, which clearly indicates the inadequacy of the current synthetic methods for producing such chiral building blocks on a large scale with sufficient environmental friendliness. See theSupporting Information(SI) for typical examples.

4. Rhodium-Catalyzed Asymmetric Addition of Aryl- and Alkenylboronic Acids to Isatins

5. Rhodium-Catalyzed Addition of Arylboronic Acids to Isatins: An Entry to Diversity in 3-Aryl-3-Hydroxyoxindoles

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