AMPA Receptor Noncompetitive Inhibitors Occupy a Promiscuous Binding Site
Author:
Affiliation:
1. Department of Chemistry, Carnegie Mellon University, Pittsburgh, Pennsylvania 15213, United States
Funder
U.S. Department of Health and Human Services
National Science Foundation
Publisher
American Chemical Society (ACS)
Subject
Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.9b00344
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5. Discovery of 2-(2-Oxo-1-phenyl-5-pyridin-2-yl-1,2-dihydropyridin-3-yl)benzonitrile (Perampanel): A Novel, Noncompetitive α-Amino-3-hydroxy-5-methyl-4-isoxazolepropanoic Acid (AMPA) Receptor Antagonist
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