Novel Highly Potent and Selective Sigma1 Receptor Antagonists Effectively Block the Binge Eating Episode in Female Rats-Reference-Cited by-同舟云学术

Novel Highly Potent and Selective Sigma1 Receptor Antagonists Effectively Block the Binge Eating Episode in Female Rats

Published:2020-09-04 Issue:19 Volume:11 Page:3107-3116
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Cifani Carlo¹^ORCID,Micioni Di Bonaventura Emanuela¹^ORCID,Botticelli Luca¹^ORCID,Del Bello Fabio²^ORCID,Giorgioni Gianfabio²^ORCID,Pavletić Pegi²,Piergentili Alessandro²^ORCID,Quaglia Wilma²^ORCID,Bonifazi Alessandro²^ORCID,Schepmann Dirk³,Wünsch Bernhard³^ORCID,Vistoli Giulio⁴^ORCID,Micioni Di Bonaventura Maria Vittoria¹^ORCID

Affiliation:

1. School of Pharmacy, Pharmacology Unit, University of Camerino, Via Madonna delle Carceri 9, 62032 Camerino, Italy

2. School of Pharmacy, Medicinal Chemistry Unit, University of Camerino, Via S. Agostino 1, 62032 Camerino, Italy

3. Institut für Pharmazeutische und Medizinische Chemie, Universität Münster, Corrensstraße 48, 48149 Münster, Germany

4. Department of Pharmaceutical Sciences, University of Milan, Via Mangiagalli 25, 20133 Milano, Italy

Funder

Universit?? degli Studi di Camerino

Ministero dell'Istruzione, dell'Universit?? e della Ricerca

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acschemneuro.0c00456

Reference57 articles.

1. Introduction to Sigma Receptors: Their Role in Disease and as Therapeutic Targets

2. Purification, molecular cloning, and expression of the mammalian sigma1-binding site.

3. Cloning and Characterization of a Mouse σ1 Receptor

4. Identification of the gene that codes for the σ2 receptor

5. Cloning and Functional Expression of the Human Type 1 Sigma Receptor (hSigmaR1)

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