Stoichiometry and Physical Chemistry of Promiscuous Aggregate-Based Inhibitors-Reference-Cited by-同舟云学术

Stoichiometry and Physical Chemistry of Promiscuous Aggregate-Based Inhibitors

Published:2008-06-28 Issue:29 Volume:130 Page:9606-9612
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Coan Kristin E. D.¹,Shoichet Brian K.¹

Affiliation:

1. Department of Pharmaceutical Chemistry & Graduate Group in Chemistry and Chemical Biology, 1700 Fourth Street, University of California at San Francisco, San Francisco, California 94158-2550

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja802977h

Reference30 articles.

1. Nonleadlikeness and leadlikeness in biochemical screening

2. Pursuing the leadlikeness concept in pharmaceutical research

3. Development of a Virtual Screening Method for Identification of “Frequent Hitters” in Compound Libraries

4. Avoiding physicochemical artefacts in early ADME–Tox experiments

5. Hit discovery and hit-to-lead approaches

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