Combination of Non-natural d-Amino Acid Derivatives and Allophenylnorstatine−Dimethylthioproline Scaffold in HIV Protease Inhibitors Have High Efficacy in Mutant HIV-Reference-Cited by-同舟云学术

Combination of Non-natural d-Amino Acid Derivatives and Allophenylnorstatine−Dimethylthioproline Scaffold in HIV Protease Inhibitors Have High Efficacy in Mutant HIV

Published:2008-04-22 Issue:10 Volume:51 Page:2992-3004
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nakatani Shingo¹,Hidaka Koushi¹,Ami Ei’ichi¹,Nakahara Koichiro¹,Sato Akihiko¹,Nguyen Jeffrey-Tri¹,Hamada Yoshio¹,Hori Yasuko¹,Ohnishi Nobuyuki¹,Nagai Akinori¹,Kimura Tooru¹,Hayashi Yoshio¹,Kiso Yoshiaki¹

Affiliation:

1. Department of Medicinal Chemistry, Center for Frontier Research in Medicinal Science, 21st Century COE Program, Kyoto Pharmaceutical University, Yamashina-ku, Kyoto 607-8412, Japan, Discovery Research Laboratories, Shionogi Co. Ltd., Settsu, Osaka 566-0022 Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm701555p

Reference36 articles.

1. UNAIDS and WHOAIDS Epidemic Update: December 2006;UNAIDS:Geneva,2006.

2. AIDS Info: A Service of the U.S. Department of Health and Human Services;http://aidsinfo.nih.gov/(accessed August 27, 2007).

3. Conserved Folding in Retroviral Proteases: Crystal Structure of Synthetic HIV-1 Protease

4. Three-dimensional structure of aspartyl protease from human immunodeficiency virus HIV-1

5. X-ray analysis of HIV-1 proteinase at 2.7 Å resolution confirms structural homology among retroviral enzymes

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