The Terminal (Catalytic) Adenosine of the HIV LTR Controls the Kinetics of Binding and Dissociation of HIV Integrase Strand Transfer Inhibitors
Author:
Affiliation:
1. Departments of Computer Assisted Drug Design, Virology, and Medicinal Chemistry, Bristol-Myers Squibb Research & Development, Wallingford, Connecticut 06492
Publisher
American Chemical Society (ACS)
Subject
Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/bi801372d
Reference47 articles.
1. Requirement of active human immunodeficiency virus type 1 integrase enzyme for productive infection of human T-lymphoid cells
2. Inhibitors of Strand Transfer That Prevent Integration and Inhibit HIV-1 Replication in Cells
3. HIV-1 integrase inhibitors that compete with the target DNA substrate define a unique strand transfer conformation for integrase
4. Integrase inhibitors to treat HIV/Aids
Cited by 40 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Brief Histories of Retroviral Integration Research and Associated International Conferences;Viruses;2024-04-13
2. Structural basis for the inhibition of HTLV-1 integration inferred from cryo-EM deltaretroviral intasome structures;Nature Communications;2021-08-17
3. Structure and function of retroviral integrase;Nature Reviews Microbiology;2021-07-09
4. Structural basis for strand-transfer inhibitor binding to HIV intasomes;Science;2020-02-14
5. Structural basis of second-generation HIV integrase inhibitor action and viral resistance;Science;2020-02-14
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3