Vinyl Sulfone-Based Peptidomimetics as Anti-Trypanosomal Agents: Design, Synthesis, Biological and Computational Evaluation-Reference-Cited by-同舟云学术

Vinyl Sulfone-Based Peptidomimetics as Anti-Trypanosomal Agents: Design, Synthesis, Biological and Computational Evaluation

Published:2013-09-03 Issue:17 Volume:56 Page:6638-6650
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Dunny Elizabeth¹,Doherty William¹,Evans Paul¹,Malthouse J. Paul G.²,Nolan Derek³,Knox Andrew J. S.³

Affiliation:

1. Centre for Synthesis and Chemical Biology, School of Chemistry and Chemical Biology, University College Dublin, Dublin 4, Ireland

2. Conway Institute, School of Biomolecular and Biomedical Science, University College Dublin, Dublin 4, Ireland

3. School of Biochemistry and Immunology, Trinity Biomedical Sciences Institute, Trinity College Dublin, Pearse Street, Dublin 2, Ireland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm400294w

Reference64 articles.

1. Drug discovery and development for neglected parasitic diseases

2. bAfrican Trypanosomiasis (Sleeping Sickness);Fact Sheet Number 259;World Health Organisation:Geneva,October 2012; http://www.who.int/mediacentre/factsheets/fS259/en/(accessed 4 December 2012).

3. Trypanosomatid Genomes

4. N-myristoyltransferase inhibitors as new leads to treat sleeping sickness

5. Cysteine Proteinase Inhibitors Kill Cultured Bloodstream Forms ofTrypanosoma brucei brucei

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