2-(3-Methyl-3H-diaziren-3-yl)ethyl 1-(1-phenylethyl)-1H-imidazole-5-carboxylate: A Derivative of the Stereoselective General Anesthetic Etomidate for Photolabeling Ligand-Gated Ion Channels-Reference-Cited by-同舟云学术

2-(3-Methyl-3H-diaziren-3-yl)ethyl 1-(1-phenylethyl)-1H-imidazole-5-carboxylate: A Derivative of the Stereoselective General Anesthetic Etomidate for Photolabeling Ligand-Gated Ion Channels

Published:2003-03-01 Issue:7 Volume:46 Page:1257-1265
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Husain S. Shaukat¹,Ziebell Michael R.¹,Ruesch Dirk¹,Hong Filbert¹,Arevalo Enrique¹,Kosterlitz Jonathan A.¹,Olsen Richard W.¹,Forman Stuart A.¹,Cohen Jonathan B.¹,Miller Keith W.¹

Affiliation:

1. Department of Anesthesia and Critical Care, Massachusetts General Hospital, Boston, Massachusetts 02114, Department of Biological Chemistry and Molecular Pharmacology and Department of Neurobiology, Harvard Medical School, Boston, Massachusetts 02115, and Department of Molecular and Medical Pharmacology, University of California School of Medicine, Los Angeles, California 90095

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020465v

Reference50 articles.

1. Anesthetics and Ion Channels: Molecular Models and Sites of Action

2. Nicotinic Receptors at the Amino Acid Level

3. Emerging structure of the Nicotinic Acetylcholine receptors

Cited by 82 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Structural interplay of anesthetics and paralytics on muscle nicotinic receptors;Nature Communications;2023-06-01

2. Pharmacological management of severe Cushing’s syndrome: the role of etomidate;Therapeutic Advances in Endocrinology and Metabolism;2022-01

3. Competitive Antagonism of Etomidate Action by Diazepam;Anesthesiology;2020-06-10

4. A potent photoreactive general anesthetic with novel binding site selectivity for GABAA receptors;European Journal of Medicinal Chemistry;2020-05

5. Allosteric GABAA Receptor Modulators—A Review on the Most Recent Heterocyclic Chemotypes and Their Synthetic Accessibility;Molecules;2020-02-24