Structure-Based Design, Synthesis, and Pharmacological Evaluation of 3-(Aminoalkyl)-5-fluoroindoles as Myeloperoxidase Inhibitors-Reference-Cited by-同舟云学术

Structure-Based Design, Synthesis, and Pharmacological Evaluation of 3-(Aminoalkyl)-5-fluoroindoles as Myeloperoxidase Inhibitors

Published:2010-11-22 Issue:24 Volume:53 Page:8747-8759
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Soubhye Jalal¹,Prévost Martine²,Van Antwerpen Pierre¹³,Zouaoui Boudjeltia Karim⁴,Rousseau Alexandre⁴,Furtmüller Paul G.⁵,Obinger Christian⁵,Vanhaeverbeek Michel⁴,Ducobu Jean⁴,Nève Jean¹,Gelbcke Michel¹,Dufrasne Franc¸ois¹

Affiliation:

1. Laboratoire de Chimie Pharmaceutique Organique, Faculté de Pharmacie, Université Libre de Bruxelles, Brussels, Belgium

2. Laboratoire de Structure et Fonction des Membranes Biologiques, Université Libre de Bruxelles, Brussels, Belgium

3. Analytical Platform of the Faculty of Pharmacy, Université Libre de Bruxelles, Brussels, Belgium

4. Laboratory of Experimental Medicine, CHU Charleroi, A. Vésale Hospital, Université Libre de Bruxelles, Montigny-le-Tilleul, Belgium

5. Department of Chemistry, Division of Biochemistry, BOKU—University of Natural Resources and Life Sciences, Vienna, Austria

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm1009988

Reference59 articles.

1. Myeloperoxidase: friend and foe

2. Myeloperoxidase and Cardiovascular Disease

3. Myeloperoxidase, modified lipoproteins, and atherogenesis

4. Neuronal expression of myeloperoxidase is increased in Alzheimer's disease

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