Design, Synthesis, and Discovery of Novel trans-Stilbene Analogues as Potent and Selective Human Cytochrome P450 1B1 Inhibitors-Reference-Cited by-同舟云学术

Design, Synthesis, and Discovery of Novel trans-Stilbene Analogues as Potent and Selective Human Cytochrome P450 1B1 Inhibitors

Published:2001-12-07 Issue:1 Volume:45 Page:160-164
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kim Sanghee¹,Ko Hyojin¹,Park Jae Eun¹,Jung Sungkyu¹,Lee Sang Kwang¹,Chun Young-Jin¹

Affiliation:

1. Natural Products Research Institute, College of Pharmacy, Seoul National University, 28 Yungun, Jongro, Seoul 110-460, Korea, and College of Pharmacy, Chungang University, 221 Huksuk, Dongjak, Seoul 156-756, Korea

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm010298j

Reference33 articles.

1. Cytochrome P450

2. Mouse endometrium stromal cells express a polycyclic aromatic hydrocarbon-inducible cytochrome P450 that closely resembles the novel P450 in mouse embryo fibroblasts (P450EF)

3. Expression of cytochrome P450 CYP1B1 in breast cancer

4. Cytochromes CYP1A1 and CYP1B1 in the rat mammary gland: Cell-specific expression and regulation by polycyclic aromatic hydrocarbons and hormones

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