Synthesis and Structure−Activity Relationships of Parasiticidal Thiosemicarbazone Cysteine Protease Inhibitors against Plasmodium falciparum, Trypanosoma brucei, and Trypanosoma cruzi-Reference-Cited by-同舟云学术

Synthesis and Structure−Activity Relationships of Parasiticidal Thiosemicarbazone Cysteine Protease Inhibitors against Plasmodium falciparum, Trypanosoma brucei, and Trypanosoma cruzi

Published:2004-05-04 Issue:12 Volume:47 Page:3212-3219
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Greenbaum Doron C.¹,Mackey Zachary¹,Hansell Elizabeth¹,Doyle Patricia¹,Gut Jiri¹,Caffrey Conor R.¹,Lehrman Julia¹,Rosenthal Philip J.¹,McKerrow James H.¹,Chibale Kelly¹

Affiliation:

1. Sandler Center for Basic Research in Parasitic Diseases, Department of Pathology, University of California, San Francisco, California 94143, Department of Medicine, San Francisco General Hospital, San Francisco, California 94143, and Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030549j

Reference18 articles.

1. Anti-HIV Activity of Thiosemicarbazone and Semicarbazone Derivatives of (±)-3-Menthone

2. A Vaccinia virus isatin-β-thiosemicarbazone resistance mutation maps in the viral gene encoding the 132-kDa subunit of RNA polymerase

3. Triapine (3-aminopyridine-2-carboxaldehyde thiosemicarbazone; 3-AP): an inhibitor of ribonucleotide reductase with antineoplastic activity

4. Analogs of methotrexate

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