Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors-Reference-Cited by-同舟云学术

Synthesis, Pharmacological Evaluation, and Molecular Modeling Studies of Novel Peptidic CAAX Analogues as Farnesyl-Protein-Transferase Inhibitors

Published:2006-02-24 Issue:6 Volume:49 Page:1882-1890
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Santagada Vincenzo¹,Caliendo Giuseppe¹,Severino Beatrice¹,Lavecchia Antonio¹,Perissutti Elisa¹,Fiorino Ferdinando¹,Zampella Angela¹,Sepe Valentina¹,Califano Daniela¹,Santelli Giovanni¹,Novellino Ettore¹

Affiliation:

1. Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli ≪Federico II≫ Via D. Montesano 49, 80131 Napoli, Italy, Dipartimento di Chimica delle Sostanze Naturali, Università di Napoli ≪Federico II≫ Via D. Montesano 49, 80131 Napoli, Italy, and Dipartimento di Oncologia Sperimentale, Istituto dei Tumori ≪Fondazione Pascale≫, via Semmola 80131, Napoli, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0506165

Reference29 articles.

1. Design, Synthesis, and Evaluation of Su- gar Amino Acid Based Inhibitors of Pro- tein Prenyl Transferases PFT and PGGT-1

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