Increased Anti-P-glycoprotein Activity of Baicalein by Alkylation on the A Ring-Reference-Cited by-同舟云学术

Increased Anti-P-glycoprotein Activity of Baicalein by Alkylation on the A Ring

Published:2004-09-22 Issue:22 Volume:47 Page:5555-5566
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lee Yashang¹,Yeo Hosup¹,Liu Shwu-Huey¹,Jiang Zaoli¹,Savizky Ruben M.¹,Austin David J.¹,Cheng Yung-chi¹

Affiliation:

1. Department of Pharmacology, Yale University School of Medicine, Department of Chemistry, Yale University, and PhytoCeutica, Inc., New Haven, Connecticut 06520

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049949c

Reference39 articles.

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2. BIOCHEMISTRY OF MULTIDRUG RESISTANCE MEDIATED BY THE MULTIDRUG TRANSPORTER

3. Cellular localization of the multidrug-resistance gene product P-glycoprotein in normal human tissues.

4. What have we learnt thus far from mice with disrupted P-glycoprotein genes?

5. Multidrug Resistance (MDR1) P-glycoprotein Enhances Esterification of Plasma Membrane Cholesterol

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