Synthesis and Biological Evaluation of 2‘-Carbamate-Linked and 2‘-Carbonate-Linked Prodrugs of Paclitaxel: Selective Activation by the Tumor-Associated Protease Plasmin-Reference-Cited by-同舟云学术

Synthesis and Biological Evaluation of 2‘-Carbamate-Linked and 2‘-Carbonate-Linked Prodrugs of Paclitaxel: Selective Activation by the Tumor-Associated Protease Plasmin

Published:2000-07-19 Issue:16 Volume:43 Page:3093-3102
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

de Groot Franciscus M. H.¹,van Berkom Leon W. A.¹,Scheeren Hans W.¹

Affiliation:

1. Department of Organic Chemistry, NSR−Center for Molecular Structure, Design and Synthesis, University of Nijmegen, Toernooiveld 1, 6525 ED Nijmegen, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0009078

Reference32 articles.

1. Stromal Cell Expression of Components of Matrix-Degrading Protease Systems in Human Cancer

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