High-Throughput Salt Screening of Synthetic Intermediates: Effects of Solvents, Counterions, and Counterion Solubility
Author:
Affiliation:
1. Product Development, Bristol-Myers Squibb Company, One Squibb Drive, New Brunswick, New Jersey 08903, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.0c00132
Reference57 articles.
1. Handbook of Pharmaceutical Salts, Properties, Selection, and Use; Stahl, P., Wermuth, C., Eds. Wiley-VCH: Weinheim, Germany, 2002; pp 1–3.
2. Lee, H. Pharmaceutical Industry Practices on Genotoxic Impurities; CRC Press, 2014; pp 404–405.
3. Salt selection for basic drugs
4. In Situ Salt Screening-A Useful Technique for Discovery Support and Preformulation Studies
5. Pharmaceutical Salts
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