Development and Manufacturing GMP Scale-Up of a Continuous Ir-Catalyzed Homogeneous Reductive Amination Reaction
Author:
Affiliation:
1. Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana 46285, United States
2. Eli Lilly SA, Dunderrow, Kinsale, Cork, Ireland
3. D&M Continuous Solutions, LLC, Greenwood, Indiana 46113, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
http://pubs.acs.org/doi/pdf/10.1021/acs.oprd.6b00148
Reference34 articles.
1. Details on the evacetrapib ACCELERATE phase III clinical trial can be found online atwww.clinicaltrials.gov.
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3. Development of a Hydrogenative Reductive Amination for the Synthesis of Evacetrapib: Unexpected Benefits of Water
4. A list of the 12 Principals of Green Chemistry may be found on the ACS website:http://www.acs.org/content/acs/en/greenchemistry/what-is-green-chemistry/principles/12-principles-of-green-chemistry.html.
5. Development and Scale-Up of a Continuous, High-Pressure, Asymmetric Hydrogenation Reaction, Workup, and Isolation
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