Preparation of the HIV Attachment Inhibitor BMS-663068. Part 3. Mechanistic Studies Enable a Scale-Independent Friedel–Crafts Acylation-Reference-Cited by-同舟云学术

Preparation of the HIV Attachment Inhibitor BMS-663068. Part 3. Mechanistic Studies Enable a Scale-Independent Friedel–Crafts Acylation

Published:2017-08-09 Issue:8 Volume:21 Page:1122-1130
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Beutner Gregory L.¹^ORCID,Albrecht Jacob¹,Fan Junying¹,Fanfair Dayne¹,Lawler Michael J.¹,Bultman Michael¹^ORCID,Chen Ke¹,Ivy Sabrina¹,Schild Richard L.¹,Tripp Jonathan C.¹,Murugesan Saravanababu¹,Dambalas Konstantinos¹,McLeod Douglas D.¹,Sweeney Jason T.¹,Eastgate Martin D.¹^ORCID,Conlon David A.¹

Affiliation:

1. Chemical & Synthetic Development, Bristol-Myers Squibb Company, One Squibb Drive, New Brunswick, New Jersey, 08903-0191, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.7b00115

Reference47 articles.

1. aLi, J. J.Heterocyclic Chemistry in Drug Discovery;Wiley:Hoboken, NJ, 2013; pp18–53.

2. Synthesis of natural products containing the pyrrolic ring

3. Structural Diversity of Organic Chemistry. A Scaffold Analysis of the CAS Registry

4. Multicomponent reactions for the synthesis of pyrroles

5. bBergman, J.; Janosik, T.InComprehensive Heterocyclic Chemistry III;Jones, G.; Ramsden, C. A., Eds.Elsevier:Amsterdam, 2008; Vol.3, pp269–351.

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