Stereoinvertive Deoxyamination of <i>trans</i>-2-Aminocyclohexanol Using Bose–Mitsunobu Azidation and Staudinger Reaction for the Stereoselective Synthesis of Edoxaban-Reference-Cited by-同舟云学术

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Stereoinvertive Deoxyamination of trans-2-Aminocyclohexanol Using Bose–Mitsunobu Azidation and Staudinger Reaction for the Stereoselective Synthesis of Edoxaban

Published:2023-08-01 Issue:8 Volume:27 Page:1517-1532
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Ochiai Hidenori¹^ORCID,Kubota Shunichi¹,Sasagawa Miwa¹,Mihara Taiki¹,Yamashita Atsuhiro²,Nakamata Tomohide²,Nishiyama Akira¹

Affiliation:

1. Pharma & Supplemental Nutrition Solutions Vehicle, Pharma Business Division, Kaneka Corporation, 1-8, Miyamae-cho, Takasago-cho, Takasago, Hyogo 676-8688, Japan

2. Ako Research and Analysis Center (ARAC), R&D Division, Osaka Synthetic Chemical Laboratories, Inc., 1325-67, Aza-Inariyama, Kizu, Ako, Hyogo 678-0165, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.3c00189

Reference45 articles.

1. Development of an Efficient Manufacturing Process for a Key Intermediate in the Synthesis of Edoxaban

2. aNagasawa, H.; Sato, K.; Yagi, T.; Kitani, Y. Process for producing thiazole derivative. WO 2005047296 A1, 2005.

3. bKawanami, K. Process for preparing compound by novel Sandmeyer-like reaction using nitroxide radical compound as reaction catalyst. WO 2012017932 A1, 2012.

4. cUeda, T. Method for producing inhibitor of activated blood coagulation factor X (FXa). WO 2015125710 A1, 2015.

5. dZhang, S.; Liu, J.; Yu, S.; Wang, P.; Jiao, X.; Wang, H. A kind of preparation method of thiazole. CN 106986883 A, 2017.

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