1. Bernstein, P. R.; Edwards, P. D.; Williams, J. C. InProgress inMedicinal Chemistry; Ellis, G. P., Luscombe, D. K., Eds.; Elsevier Science: New York, 1994; Vol. 31, p 59. Edwards, P. D.; Bernstein, P. R.Med. Res.Rev.1994,14, 127. Powers, J. C.; Harper, J. W. InProteinase Inhibitors; Barrett, A. J., Salvesen, G., Eds.; Elsevier Science: New York, 1986; pp 55−141.
2. Inhibition of serine proteases by peptidyl fluoromethyl ketones
3. Use of peptide aldehydes to generate transition-state analogs of elastase
4. Peptidyl carbamates incorporating amino acid isosteres as novel elastase inhibitors