Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus

Author:

Klug Dana M.1,Tse Edwin G.1,Silva Daniel G.12ORCID,Cao Yafeng3,Charman Susan A.4ORCID,Chauhan Jyoti5ORCID,Crighton Elly4,Dichiara Maria5,Drake Chris6,Drewry David78ORCID,da Silva Emery Flavio2ORCID,Ferrins Lori5ORCID,Graves Lee9ORCID,Hopkins Emily6,Kresina Thomas A. C.5,Lorente-Macías Álvaro91011ORCID,Perry Benjamin12ORCID,Phipps Richard6,Quiroga Bruno5,Quotadamo Antonio513,Sabatino Giada N.1ORCID,Sama Anthony14,Schätzlein Andreas1ORCID,Simpson Quillon J.5,Steele Jonathan6,Shanu-Wilson Julia6,Sjö Peter12,Stapleton Paul1,Swain Christopher J.15ORCID,Vaideanu Alexandra1ORCID,Xie Huanxu3,Zuercher William7ORCID,Todd Matthew H.116ORCID

Affiliation:

1. School of Pharmacy, University College London, 29-39 Brunswick Square, London WC1N 1AX, United Kingdom

2. School of Pharmaceutical Sciences of Ribeirão Preto, University of São Paulo, Ribeirão Preto, São Paulo 14040-903. Brazil

3. WuXi AppTec (Wuhan) Co., Ltd., 666 Gaoxin Road, East Lake High-Tech Development Zone, Wuhan 430075, People’s Republic of China

4. Centre for Drug Candidate Optimization, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC 3052, Australia

5. Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, United States

6. Hypha Discovery, 154b Brook Dr, Milton, Abingdon OX14 4SD, United Kingdom

7. UNC Lineberger Comprehensive Cancer Center, School of Medicine, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina 27599, United States

8. Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina 27599, United States

9. Department of Pharmacology, University of North Carolina at Chapel Hill, Chapel Hill, North Carolina 27599, United States

10. Department of Medicinal & Organic Chemistry and Excellence Research Unit of ‘‘Chemistry Applied to Biomedicine and the Environment’’, Faculty of Pharmacy, University of Granada, Campus de Cartuja s/n, 18071 Granada, Spain

11. A. L-M. Cancer Research UK Edinburgh Centre, Institute of Genetics & Cancer, University of Edinburgh, Edinburgh EH4 2XR, United Kingdom

12. Drugs for Neglected Diseases initiative (DNDi), 15 Chemin Camille-Vidart, 1202 Geneva, Switzerland

13. Clinical and Experimental Medicine PhD Program, University of Modena and Reggio Emilia, 41121 Modena, Italy

14. Citizen scientist, New York, New York 11570, United States

15. Cambridge MedChem Consulting, 8 Mangers Lane, Duxford, Cambridge CB22 4RN, United Kingdom

16. Structural Genomics Consortium, University College London, 29-39 Brunswick Square, London WC1N 1AX, United Kingdom

Funder

Monash University

University of North Carolina at Chapel Hill

National Institute of Allergy and Infectious Diseases

Direktion f?r Entwicklung und Zusammenarbeit

Agence Fran?aise de D?veloppement

M?decins Sans Fronti?res

Foreign, Commonwealth and Development Office

Ministerio de Educaci?n, Cultura y Deporte

Funda??o de Amparo ? Pesquisa do Estado de S?o Paulo

University College London

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

Reference41 articles.

Cited by 2 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3