Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors

Author:

Landi Giacomo1,Linciano Pasquale2,Borsari Chiara2,Bertolacini Claudia P.3,Moraes Carolina B.3,Cordeiro-da-Silva Anabela4,Gul Sheraz5,Witt Gesa5,Kuzikov Maria5,Costi Maria Paola2ORCID,Pozzi Cecilia1ORCID,Mangani Stefano1ORCID

Affiliation:

1. Department of Biotechnology, Chemistry and Pharmacy—Department of Excellence 2018−2020, University of Siena, via Aldo Moro 2, 53100 Siena, Italy

2. Department of Life Science, University of Modena and Reggio Emilia, via Campi 103, 41125 Modena, Italy

3. National Laboratory of Biosciences, National Center for Research in Energy and Materials, Campinas, São Paulo 13083-970, Brazil

4. Instituto de Investigação e Inovação em Saúde and IBMC-Institute for Molecular and Cell Biology, Universidade do Porto and Departamento de Ciências Biológicas, Faculdade de Farmácia da Universidade do Porto (FFUP), 4150-180 Porto, Portugal

5. Fraunhofer Institute for Molecular Biology & Applied Ecology—ScreeningPort, Schnackenburgallee 114, D-22525 Hamburg, Germany

Funder

FP7 Health

Publisher

American Chemical Society (ACS)

Subject

Infectious Diseases

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