Discovery of 1-(4-Fluorophenyl)-(3R)-[3-(4-fluorophenyl)-(3S)- hydroxypropyl]-(4S)-(4-hydroxyphenyl)-2-azetidinone (SCH 58235): A Designed, Potent, Orally Active Inhibitor of Cholesterol Absorption-Reference-Cited by-同舟云学术

Discovery of 1-(4-Fluorophenyl)-(3R)-[3-(4-fluorophenyl)-(3S)- hydroxypropyl]-(4S)-(4-hydroxyphenyl)-2-azetidinone (SCH 58235): A Designed, Potent, Orally Active Inhibitor of Cholesterol Absorption

Published:1998-02-14 Issue:6 Volume:41 Page:973-980
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rosenblum Stuart B.¹,Huynh Tram¹,Afonso Adriano¹,Davis Harry R.¹,Yumibe Nathan¹,Clader John W.¹,Burnett Duane A.¹

Affiliation:

1. Department of Discovery Research, Schering-Plough Research Institute, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033-0539

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970701f

Reference23 articles.

1. Section Review—Cardiovascular & Renal: Emerging Therapies in Atherosclerosis

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