A Peptide-Based Biosensor Assay To Detect Intracellular Syk Kinase Activation and Inhibition
Author:
Affiliation:
1. Department of Medicinal Chemistry and Molecular Pharmacology and Purdue Center for Cancer Research, Purdue University, West Lafayette, Indiana 47907, United States
Publisher
American Chemical Society (ACS)
Subject
Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/bi300970h
Reference47 articles.
1. Purification and characterization of a cytosolic protein-tyrosine kinase from porcine spleen
2. Purification and characterization of a protein-tyrosine kinase from bovine thymus.
3. Perinatal lethality and blocked B-cell development in mice lacking the tyrosine kinase Syk
4. Specific Inhibition of Spleen Tyrosine Kinase Suppresses Leukocyte Immune Function and Inflammation in Animal Models of Rheumatoid Arthritis
5. A novel Syk family kinase inhibitor: Design, synthesis, and structure–activity relationship of 1,2,4-triazolo[4,3-c]pyrimidine and 1,2,4-triazolo[1,5-c]pyrimidine derivatives
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