Design and Microwave-Assisted Synthesis of Novel Macrocyclic Peptides Active at Melanocortin Receptors: Discovery of Potent and Selective hMC5R Receptor Antagonists-Reference-Cited by-同舟云学术

Design and Microwave-Assisted Synthesis of Novel Macrocyclic Peptides Active at Melanocortin Receptors: Discovery of Potent and Selective hMC5R Receptor Antagonists

Published:2008-04-15 Issue:9 Volume:51 Page:2701-2707
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Grieco Paolo¹,Cai Minying¹,Liu Lu¹,Mayorov Alexander¹,Chandler Kevin¹,Trivedi Dev¹,Lin Guangxin¹,Campiglia Pietro¹,Novellino Ettore¹,Hruby Victor J.¹

Affiliation:

1. Department of Chemistry, University of Arizona, Tucson, Arizona 85721, Department of Pharmaceutical Chemistry and Toxicology, University of Napoli “Federico II”, Naples, Italy, and Department of Pharmaceutical Science, University of Salerno, Fisciano, Salerno, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm701181n

Reference66 articles.

1. Biosynthesis of adrenocorticotropic hormone in mouse pituitary tumor cells.

2. Structure and Biosynthesis of Pro-Adrenocorticotropin/Endorphin and Related Peptides*

3. Regulation of the Synthesis of Steroidogenic Enzymes in Adrenal Cortical Cells by ACTH

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