Potent, Small-Molecule Inhibitors of Human Mast Cell Tryptase. Antiasthmatic Action of a Dipeptide-Based Transition-State Analogue Containing a Benzothiazole Ketone-Reference-Cited by-同舟云学术

Potent, Small-Molecule Inhibitors of Human Mast Cell Tryptase. Antiasthmatic Action of a Dipeptide-Based Transition-State Analogue Containing a Benzothiazole Ketone

Published:2003-08-01 Issue:18 Volume:46 Page:3865-3876
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Costanzo Michael J.¹,Yabut Stephen C.¹,Almond, Harold R.¹,Andrade-Gordon Patricia¹,Corcoran Thomas W.¹,de Garavilla Lawrence¹,Kauffman Jack A.¹,Abraham William M.¹,Recacha Rosario¹,Chattopadhyay Debashish¹,Maryanoff Bruce E.¹

Affiliation:

1. Drug Discovery, Johnson & Johnson Pharmaceutical Research & Development, Spring House, Pennsylvania 19477-0776, Division of Pulmonary Disease, University of Miami at Mount Sinai Medical Center, Miami Beach, Florida 33140, and Centre for Macromolecular Studies, University of Alabama at Birmingham, Birmingham, Alabama 35294

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030050p

Reference39 articles.

1. Of mites and men: trypsin-like proteases in the lungs.

2. [7] Hepsin

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