Allosteric Modulation of the Adenosine A1 Receptor. Synthesis and Biological Evaluation of Novel 2-Amino-3-benzoylthiophenes as Allosteric Enhancers of Agonist Binding-Reference-Cited by-同舟云学术

Allosteric Modulation of the Adenosine A1 Receptor. Synthesis and Biological Evaluation of Novel 2-Amino-3-benzoylthiophenes as Allosteric Enhancers of Agonist Binding

Published:1999-08-19 Issue:18 Volume:42 Page:3629-3635
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

van der Klein Pieter A. M.¹,Kourounakis Angeliki P.¹,IJzerman Ad P.¹

Affiliation:

1. Division of Medicinal Chemistry, Leiden/Amsterdam Center for Drug Research, P.O. Box 9502, 2300 RA Leiden, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm991051d

Reference31 articles.

1. Jacobson, K. A.; van Rhee, A. M. Development of selective purinoceptor agonists and antagonists.Purinergicapproachesinexperimentaltherapeutics; Jacobson, K. A., Jarvis, M. F., Eds.; Wiley-Liss: New York, 1997; pp 101−128.

2. Stiles, G. L. Adenosine receptor subtypes: new insights from cloning and functional studies.Purinergicapproachesinexperimentaltherapeutics; Jacobson, K. A., Jarvis, M. F., Eds.; Wiley-Liss: New York, 1997; pp 29−37.

Cited by 94 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Truly Catalytic Gewald Synthesis of 2-Aminothiophenes Using Piperidinium Borate (Pip Borate), a Conjugate Acid–Base Pair;SynOpen;2023-10-10

2. Small molecule allosteric modulation of the adenosine A1 receptor;Frontiers in Endocrinology;2023-06-26

3. Allosteric Modulators of Adenosine Receptors;Topics in Medicinal Chemistry;2022

4. Multisite Model of Allosterism for the Adenosine A1 Receptor;Journal of Chemical Information and Modeling;2021-03-29

5. A Multisite Model of Allosterism for the Adenosine A1 Receptor;2020-10-14