N,N′-Carbonyldiimidazole-Mediated Amide Coupling: Significant Rate Enhancement Achieved by Acid Catalysis with Imidazole·HCl
Author:
Affiliation:
1. AstraZeneca, Global PR&D, Avlon Works, Severn Road, Hallen, Bristol BS10 7ZE, U.K.
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/op800226b
Reference28 articles.
1. Amide bond formation and peptide coupling
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3. The Chemical Development of the Commercial Route to Sildenafil: A Case History
4. Carbamoylimidazolium and thiocarbamoylimidazolium salts: novel reagents for the synthesis of ureas, thioureas, carbamates, thiocarbamates and amides
5. Amidations Using N,N ‘-Carbonyldiimidazole: Remarkable Rate Enhancement by Carbon Dioxide
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